CB1R antagonist 1( —— )

Catalog No. M35611 CAS No. 334668-69-8

CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

CB1R antagonist 1
Note

Research use only, not for human use.
Brief Description

CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.
Description

CB1R Allosteric modulator 5, a selective cannabinoid-1 receptor (CB1R) inverse agonist with an IC50 value of 4.2 μM and EC50 value of ＞10 μM. CB1R Allosteric modulator 5 can be used for the research of metabolic and obesity.
In Vitro

CB1R Allosteric modulator 5 has cannabinoid-1 receptor (CB1R) activity with an IC50value of 4.2 μM and EC50 value of ＞10 μM.
In Vivo

——
Synonyms

——
Pathway

GPCR/G Protein
Target

Cannabinoid Receptor
Recptor

Cannabinoid Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

334668-69-8
Formula Weight

404.45
Molecular Formula

C18H23F3N2O3S
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 100 mg/mL (247.25 mM; Ultrasonic )
SMILES

S(=O)(=O)(C1=CC(C(F)(F)F)=CC=C1)N2CCN(C(=O)C3CCCCC3)CC2
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Petr Vachal, et al. 1-Sulfonyl-4-acylpiperazines as selective cannabinoid-1 receptor (CB1R) inverse agonists for the treatment of obesity. J Med Chem. 2009 Apr 23;52(8):2550-8?

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